Acefurtiamine
Chemical compound
- none
- (3E)-4-{[(4-Amino-2-methylpyrimidin-5-yl)methyl](formyl)amino}-3-[(furan-2-ylcarbonyl)sulfanyl]pent-3-en-1-yl (acetyloxy)acetate
- 10072-48-7 N
- 3037171
- 2300987 Y
- 6APJ3D1308
- ChEMBL2104090 N
- DTXSID20864202
- Interactive image
- O=C(OCC(=O)OCCC(\SC(=O)c1occc1)=C(/N(C=O)Cc2cnc(nc2N)C)C)C
InChI
- InChI=1S/C21H24N4O7S/c1-13(25(12-26)10-16-9-23-14(2)24-20(16)22)18(33-21(29)17-5-4-7-30-17)6-8-31-19(28)11-32-15(3)27/h4-5,7,9,12H,6,8,10-11H2,1-3H3,(H2,22,23,24)/b18-13+ Y
- Key:MYBUGVXNAHWTOL-QGOAFFKASA-N Y
Acefurtiamine (INN) is a vitamin B1 analog in a manner similar to the GABAergic activity of the thiamine derivative clomethiazole.[1] It functions as an analgesic agent at sufficient doses.[medical citation needed]
References
- ^ Martindale W (1993). The Extra Pharmacopoeia. Pharmaceutical Press. p. 1053. ISBN 978-0-85369-300-0.
Further reading
- Elks J, Ganellin CR, eds. (1990). The Dictionary of Drugs: Chemical Data: Chemical Data, Structures and Bibliographies. Springer. pp. 2–. doi:10.1007/978-1-4757-2085-3. ISBN 978-1-4757-2085-3.
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Vitamins (A11)
soluble
A | |
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D | |
E | |
K |
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soluble
B |
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C |
- #WHO-EM
- ‡Withdrawn from market
- Clinical trials:
- †Phase III
- §Never to phase III
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